Basic Peptide Information

DICL ID
DICL_Pep_06951
Ion Channel
Neuronal acetylcholine receptor subunit alpha-7
Peptide Function
Antagonist
Gene Name
CHRNA7

Activity Data (nM)

IC50
23 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified

Sequence Information

Peptide Sequence
GPCSCGHGRRWHYVCTCGNRPCC(Nle)SGC(Nle)RTRC
Peptide UniProt Accession
Not available
UniParc
Not available
Peptide Synonyms/Alias
VxXXB CTD(19–50)
Peptide Species
Not specified
Peptide Name
Not available
CAS Number
Not available

Experimental Conditions

pH
Not mention
Holding Potential (mV)
Not specified
Temperature
Not mention
Test Method
Fluorescence assay
Test Species
SH-SY5Y neuroblastoma cell

Binding Information

Binding Site
Not specified
Binding Site Residue
Not specified

Ion Channel Information

Gene Abbreviation (ABB)
nAChRs
Ion Channel UniProt Accession
Source Organism
Homo sapiens (Human)

References & Disease Information

Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available